CAS RN 1309198-71-7
CAS RN 1309198-71-7
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Tocris Bioscience™ Ogerin
Selective positive allosteric modulator at GPR68
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Ogerin, MedChemExpress
MedChemExpress Ogerin is a selective GPR68 positive allosteric modulator, with a pEC50 of 6.83. Ogerin shows inverse agonist and antagonist activity (Ki, 220 nM) at A2A receptoor and weak antagonist activity (Ki, 736 nM) at 5-HT2B receptor. Ogerin blocks recall in fear conditioning in mice.
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